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Professor Christian Sergheraert

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    Publications listed below are automatically derived from MEDLINE/PubMed and other sources, which might result in incorrect or missing publications. Faculty can login to make corrections and additions.
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    1. Melnyk P, Vingtdeux V, Burlet S, Eddarkaoui S, Grosjean ME, Larchanché PE, Hochart G, Sergheraert C, Estrella C, Barrier M, Poix V, Plancq P, Lannoo C, Hamdane M, Delacourte A, Verwaerde P, Buée L, Sergeant N. Chloroquine and chloroquinoline derivatives as models for the design of modulators of amyloid Peptide precursor metabolism. ACS Chem Neurosci. 2015 Apr 15; 6(4):559-69. PMID: 25611616.
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    2. Delarue-Cochin S, Grellier P, Maes L, Mouray E, Sergheraert C, Melnyk P. Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline. Eur J Med Chem. 2008 Oct; 43(10):2045-55. PMID: 18226428.
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    3. Delarue-Cochin S, Paunescu E, Maes L, Mouray E, Sergheraert C, Grellier P, Melnyk P. Synthesis and antimalarial activity of new analogues of amodiaquine. Eur J Med Chem. 2008 Feb; 43(2):252-60. PMID: 17485145.
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    4. Mouray E, Moutiez M, Girault S, Sergheraert C, Florent I, Grellier P. Biochemical properties and cellular localization of Plasmodium falciparum protein disulfide isomerase. Biochimie. 2007 Mar; 89(3):337-46. PMID: 17166645.
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    5. Helleboid-Chapman A, Helleboid S, Jakel H, Timmerman C, Sergheraert C, Pattou F, Fruchart-Najib J, Fruchart JC. Glucose regulates LXRalpha subcellular localization and function in rat pancreatic beta-cells. Cell Res. 2006 Jul; 16(7):661-70. PMID: 16773041.
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    6. Charton J, Girault-Mizzi S, Debreu-Fontaine MA, Foufelle F, Hainault I, Bizot-Espiard JG, Caignard DH, Sergheraert C. Synthesis and biological evaluation of benzimidazole derivatives as potent AMP-activated protein kinase activators. Bioorg Med Chem. 2006 Jul 01; 14(13):4490-518. PMID: 16513356.
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    7. Melnyk P, Leroux V, Sergheraert C, Grellier P. Design, synthesis and in vitro antimalarial activity of an acylhydrazone library. Bioorg Med Chem Lett. 2006 Jan 01; 16(1):31-5. PMID: 16263280.
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    8. Charton J, Cazenave Gassiot A, Girault-Mizzi S, Debreu-Fontaine MA, Melnyk P, Sergheraert C. Synthesis and pharmacological evaluation of Tic-hydantoin derivatives as selective sigma1 ligands. Part 1. Bioorg Med Chem Lett. 2005 Nov 01; 15(21):4833-7. PMID: 16140011.
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    9. Cazenave Gassiot A, Charton J, Girault-Mizzi S, Gilleron P, Debreu-Fontaine MA, Sergheraert C, Melnyk P. Synthesis and pharmacological evaluation of Tic-hydantoin derivatives as selective sigma1 ligands. Part 2. Bioorg Med Chem Lett. 2005 Nov 01; 15(21):4828-32. PMID: 16140009.
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    10. Ryckebusch A, Gilleron P, Millet R, Houssin R, Lemoine A, Pommery N, Grellier P, Sergheraert C, Hénichart JP. Novel N-(4-Piperidinyl)benzamide antimalarials with mammalian protein farnesyltransferase inhibitory activity. Chem Pharm Bull (Tokyo). 2005 Oct; 53(10):1324-6. PMID: 16204993.
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    11. Charton J, Girault-Mizzi S, Sergheraert C. Conversion of sterically hindered diacylated 1,2-phenylenediamines into 2-substituted benzimidazoles. Chem Pharm Bull (Tokyo). 2005 May; 53(5):492-7. PMID: 15863918.
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    12. Ryckebusch A, Debreu-Fontaine MA, Mouray E, Grellier P, Sergheraert C, Melnyk P. Synthesis and antimalarial evaluation of new N1-(7-chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine derivatives. Bioorg Med Chem Lett. 2005 Jan 17; 15(2):297-302. PMID: 15603943.
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    13. Ryckebusch A, Fruchart JS, Cattiaux L, Rousselot-Paillet P, Leroux V, Melnyk O, Grellier P, Mouray E, Sergheraert C, Melnyk P. Design, synthesis and antimalarial activity of a glyoxylylhydrazone library. Bioorg Med Chem Lett. 2004 Sep 06; 14(17):4439-43. PMID: 15357968.
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    14. Temmerman S, Pethe K, Parra M, Alonso S, Rouanet C, Pickett T, Drowart A, Debrie AS, Delogu G, Menozzi FD, Sergheraert C, Brennan MJ, Mascart F, Locht C. Methylation-dependent T cell immunity to Mycobacterium tuberculosis heparin-binding hemagglutinin. Nat Med. 2004 Sep; 10(9):935-41. PMID: 15300244.
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    15. Guillon J, Grellier P, Labaied M, Sonnet P, Léger JM, Déprez-Poulain R, Forfar-Bares I, Dallemagne P, Lemaître N, Péhourcq F, Rochette J, Sergheraert C, Jarry C. Synthesis, antimalarial activity, and molecular modeling of new pyrrolo[1,2-a]quinoxalines, bispyrrolo[1,2-a]quinoxalines, bispyrido[3,2-e]pyrrolo[1,2-a]pyrazines, and bispyrrolo[1,2-a]thieno[3,2-e]pyrazines. J Med Chem. 2004 Apr 08; 47(8):1997-2009. PMID: 15055999.
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    16. Soulère L, Delplace P, Davioud-Charvet E, Py S, Sergheraert C, Périé J, Ricard I, Hoffmann P, Dive D. Screening of Plasmodium falciparum iron superoxide dismutase inhibitors and accuracy of the SOD-assays. Bioorg Med Chem. 2003 Nov 17; 11(23):4941-4. PMID: 14604655.
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    17. Ryckebusch A, Deprez-Poulain R, Debreu-Fontaine MA, Vandaele R, Mouray E, Grellier P, Sergheraert C. Synthesis and antimalarial evaluation of new 1,4-bis(3-aminopropyl)piperazine derivatives. Bioorg Med Chem Lett. 2003 Nov 03; 13(21):3783-7. PMID: 14552779.
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    18. Flipo M, Florent I, Grellier P, Sergheraert C, Deprez-Poulain R. Design, synthesis and antimalarial activity of novel, quinoline-based, zinc metallo-aminopeptidase inhibitors. Bioorg Med Chem Lett. 2003 Aug 18; 13(16):2659-62. PMID: 12873488.
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    19. Sergeant N, Bombois S, Ghestem A, Drobecq H, Kostanjevecki V, Missiaen C, Wattez A, David JP, Vanmechelen E, Sergheraert C, Delacourte A. Truncated beta-amyloid peptide species in pre-clinical Alzheimer's disease as new targets for the vaccination approach. J Neurochem. 2003 Jun; 85(6):1581-91. PMID: 12787077.
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    20. Rousseaux-Prévost R, Lécuyer C, Drobecq H, Sergheraert C, Dacheux JL, Rousseaux J. Characterization of boar sperm cytoskeletal cylicin II as an actin-binding protein. Biochem Biophys Res Commun. 2003 Mar 28; 303(1):182-9. PMID: 12646184.
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    21. Ryckebusch A, Deprez-Poulain R, Maes L, Debreu-Fontaine MA, Mouray E, Grellier P, Sergheraert C. Synthesis and in vitro and in vivo antimalarial activity of N1-(7-chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine derivatives. J Med Chem. 2003 Feb 13; 46(4):542-57. PMID: 12570376.
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    22. Millet R, Maes L, Landry V, Sergheraert C, Davioud-Charvet E. Antitrypanosomal activities and cytotoxicity of 5-nitro-2-furancarbohydrazides. Bioorg Med Chem Lett. 2002 Dec 16; 12(24):3601-4. PMID: 12443785.
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    23. Ryckebusch A, Déprez-Poulain R, Debreu-Fontaine MA, Vandaele R, Mouray E, Grellier P, Sergheraert C. Parallel synthesis and anti-malarial activity of a sulfonamide library. Bioorg Med Chem Lett. 2002 Sep 16; 12(18):2595-8. PMID: 12182868.
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    24. Pethe K, Bifani P, Drobecq H, Sergheraert C, Debrie AS, Locht C, Menozzi FD. Mycobacterial heparin-binding hemagglutinin and laminin-binding protein share antigenic methyllysines that confer resistance to proteolysis. Proc Natl Acad Sci U S A. 2002 Aug 06; 99(16):10759-64. PMID: 12149464.
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    25. Vendeville S, Goossens F, Debreu-Fontaine MA, Landry V, Davioud-Charvet E, Grellier P, Scharpe S, Sergheraert C. Comparison of the inhibition of human and Trypanosoma cruzi prolyl endopeptidases. Bioorg Med Chem. 2002 Jun; 10(6):1719-29. PMID: 11937331.
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    26. Davioud-Charvet E, Delarue S, Biot C, Schwöbel B, Boehme CC, Müssigbrodt A, Maes L, Sergheraert C, Grellier P, Schirmer RH, Becker K. A prodrug form of a Plasmodium falciparum glutathione reductase inhibitor conjugated with a 4-anilinoquinoline. J Med Chem. 2001 Nov 22; 44(24):4268-76. PMID: 11708927.
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    27. Grellier P, Vendeville S, Joyeau R, Bastos IM, Drobecq H, Frappier F, Teixeira AR, Schrével J, Davioud-Charvet E, Sergheraert C, Santana JM. Trypanosoma cruzi prolyl oligopeptidase Tc80 is involved in nonphagocytic mammalian cell invasion by trypomastigotes. J Biol Chem. 2001 Dec 14; 276(50):47078-86. PMID: 11598112.
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    28. Delarue S, Girault S, Maes L, Debreu-Fontaine MA, Labaeïd M, Grellier P, Sergheraert C. Synthesis and in vitro and in vivo antimalarial activity of new 4-anilinoquinolines. J Med Chem. 2001 Aug 16; 44(17):2827-33. PMID: 11495593.
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    29. Delarue S, Girault S, Dali Ali F, Maes L, Grellier P, Sergheraert C. "One-pot" synthesis and antimalarial activity of formamidine derivatives of 4-anilinoquinoline. Chem Pharm Bull (Tokyo). 2001 Aug; 49(8):933-7. PMID: 11515580.
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    30. Xu KP, Zoukhri D, Zieske JD, Dartt DA, Sergheraert C, Loing E, Yu FS. A role for MAP kinase in regulating ectodomain shedding of APLP2 in corneal epithelial cells. Am J Physiol Cell Physiol. 2001 Aug; 281(2):C603-14. PMID: 11443060.
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    31. Girault S, Delarue S, Grellier P, Berecibar A, Maes L, Quirijnen L, Lemiere P, Debreu-Fontaine MA, Sergheraert C. Antimalarial in-vivo activity of bis(9-amino-6-chloro-2-methoxyacridines). J Pharm Pharmacol. 2001 Jul; 53(7):935-8. PMID: 11480542.
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    32. Girault S, Grellier P, Berecibar A, Maes L, Lemière P, Mouray E, Davioud-Charvet E, Sergheraert C. Antiplasmodial activity and cytotoxicity of bis-, tris-, and tetraquinolines with linear or cyclic amino linkers. J Med Chem. 2001 May 24; 44(11):1658-65. PMID: 11356101.
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    33. Girault S, Davioud-Charvet TE, Maes L, Dubremetz JF, Debreu MA, Landry V, Sergheraert C. Potent and specific inhibitors of trypanothione reductase from Trypanosoma cruzi: bis(2-aminodiphenylsulfides) for fluorescent labeling studies. Bioorg Med Chem. 2001 Apr; 9(4):837-46. PMID: 11354666.
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    34. Matias I, Bisogno T, Melck D, Vandenbulcke F, Verger-Bocquet M, De Petrocellis L, Sergheraert C, Breton C, Di Marzo V, Salzet M. Evidence for an endocannabinoid system in the central nervous system of the leech Hirudo medicinalis. Brain Res Mol Brain Res. 2001 Mar 05; 87(2):145-59. PMID: 11245916.
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    35. Salmon-Chemin L, Buisine E, Yardley V, Kohler S, Debreu MA, Landry V, Sergheraert C, Croft SL, Krauth-Siegel RL, Davioud-Charvet E. 2- and 3-substituted 1,4-naphthoquinone derivatives as subversive substrates of trypanothione reductase and lipoamide dehydrogenase from Trypanosoma cruzi: synthesis and correlation between redox cycling activities and in vitro cytotoxicity. J Med Chem. 2001 Feb 15; 44(4):548-65. PMID: 11170645.
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    36. Florent I, Mouray E, Dali Ali F, Drobecq H, Girault S, Schrével J, Sergheraert C, Grellier P, Florenta I. Cloning of Plasmodium falciparum protein disulfide isomerase homologue by affinity purification using the antiplasmodial inhibitor 1,4-bis[3-[N-(cyclohexyl methyl)amino]propyl]piperazine.. FEBS Lett. 2000 Nov 10; 484(3):246-52. PMID: 11078887.
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    37. Girault S, Grellier P, Berecibar A, Maes L, Mouray E, Lemière P, Debreu MA, Davioud-Charvet E, Sergheraert C. Antimalarial, antitrypanosomal, and antileishmanial activities and cytotoxicity of bis(9-amino-6-chloro-2-methoxyacridines): influence of the linker. J Med Chem. 2000 Jul 13; 43(14):2646-54. PMID: 10893302.
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    38. Salmon-Chemin L, Lemaire A, De Freitas S, Deprez B, Sergheraert C, Davioud-Charvet E. Parallel synthesis of a library of 1,4-naphthoquinones and automated screening of potential inhibitors of trypanothione reductase from Trypanosoma cruzi. Bioorg Med Chem Lett. 2000 Apr 03; 10(7):631-5. PMID: 10762041.
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    39. Zoukhri D, Hodges RR, Sergheraert C, Dartt DA. Cholinergic-induced Ca2+ elevation in rat lacrimal gland acini is negatively modulated by PKCdelta and PKCepsilon. Invest Ophthalmol Vis Sci. 2000 Feb; 41(2):386-92. PMID: 10670466.
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    40. Bonnet B, Soullez D, Girault S, Maes L, Landry V, Davioud-Charvet E, Sergheraert C. Trypanothione reductase inhibition/trypanocidal activity relationships in a 1,4-bis(3-aminopropyl)piperazine series. Bioorg Med Chem. 2000 Jan; 8(1):95-103. PMID: 10968268.
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    41. Choukhi A, Pillez A, Drobecq H, Sergheraert C, Wychowski C, Dubuisson J. Characterization of aggregates of hepatitis C virus glycoproteins. J Gen Virol. 1999 Dec; 80 ( Pt 12):3099-3107. PMID: 10567640.
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    42. Thiam K, Loing E, Zoukhri D, Rommens C, Hodges R, Dartt D, Verwaerde C, Auriault C, Gras-Masse H, Sergheraert C. Direct evidence of cytoplasmic delivery of PKC-alpha, -epsilon and -zeta pseudosubstrate lipopeptides: study of their implication in the induction of apoptosis. FEBS Lett. 1999 Oct 15; 459(3):285-90. PMID: 10526151.
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    43. Davioud-Charvet E, Berecibar A, Girault S, Landry V, Drobecq H, Sergheraert C. Synthesis of polyamine derivatives for the preparation of affinity chromatography columns for the search of new Trypanosoma cruzi targets. Bioorg Med Chem Lett. 1999 Jun 07; 9(11):1567-72. PMID: 10386937.
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    44. Davioud-Charvet E, Becker K, Landry V, Gromer S, Logé C, Sergheraert C. Synthesis of 5,5'-dithiobis(2-nitrobenzamides) as alternative substrates for trypanothione reductase and thioredoxin reductase: a microtiter colorimetric assay for inhibitor screening. Anal Biochem. 1999 Mar 01; 268(1):1-8. PMID: 10036154.
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    45. Vendeville S, Bourel L, Davioud-Charvet E, Grellier P, Deprez B, Sergheraert C. Automated parallel synthesis of a tetrahydroisoquinolin-based library: potential prolyl endopeptidase inhibitors. Bioorg Med Chem Lett. 1999 Feb 08; 9(3):437-42. PMID: 10091698.
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    46. Vendeville S, Buisine E, Williard X, Schrevel J, Grellier P, Santana J, Sergheraert C. Identification of inhibitors of an 80 kDa protease from Trypanosoma cruzi through the screening of a combinatorial peptide library. Chem Pharm Bull (Tokyo). 1999 Feb; 47(2):194-8. PMID: 10071854.
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    47. Girault S, Davioud-Charvet E, Salmon L, Berecibar A, Debreu MA, Sergheraert C. Structure-activity relationships in 2-aminodiphenylsulfides against trypanothione reductase from Trypanosoma cruzi. Bioorg Med Chem Lett. 1998 May 19; 8(10):1175-80. PMID: 9871730.
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    48. Zoukhri D, Hodges RR, Sergheraert C, Dartt DA. Lacrimal gland functions are differentially controlled by protein kinase C isoforms. Ann N Y Acad Sci. 1998 Apr 15; 842:217-20. PMID: 9599315.
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    49. Salmon L, Landry V, Melnyk O, Maes L, Sergheraert C, Davioud-Charvet E. A general approach to the synthesis of polyamine linked-monoindolylmaleimides, a new series of trypanothione reductase inhibitors. Chem Pharm Bull (Tokyo). 1998 Apr; 46(4):707-10. PMID: 9579046.
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    50. Zoukhri D, Hodges RR, Sergheraert C, Dartt DA. Protein kinase C isoforms differentially control lacrimal gland functions. Adv Exp Med Biol. 1998; 438:181-6. PMID: 9634884.
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    51. Bonnet B, Soullez D, Davioud-Charvet E, Landry V, Horvath D, Sergheraert C. New spermine and spermidine derivatives as potent inhibitors of Trypanosoma cruzi trypanothione reductase. Bioorg Med Chem. 1997 Jul; 5(7):1249-56. PMID: 9377084.
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    52. Sohn UD, Zoukhri D, Dartt D, Sergheraert C, Harnett KM, Behar J, Biancani P. Different protein kinase C isozymes mediate lower esophageal sphincter tone and phasic contraction of esophageal circular smooth muscle. Mol Pharmacol. 1997 Mar; 51(3):462-70. PMID: 9058601.
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    53. Hodges RR, Zoukhri D, Sergheraert C, Zieske JD, Dartt DA. Identification of vasoactive intestinal peptide receptor subtypes in the lacrimal gland and their signal-transducing components. Invest Ophthalmol Vis Sci. 1997 Mar; 38(3):610-9. PMID: 9071214.
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    54. Gonindard C, Bergonzi C, Denier C, Sergheraert C, Klaebe A, Chavant L, Hollande E. Synthetic hispidin, a PKC inhibitor, is more cytotoxic toward cancer cells than normal cells in vitro. Cell Biol Toxicol. 1997 Mar; 13(3):141-53. PMID: 9088624.
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    55. Moutiez M, Quéméneur E, Sergheraert C, Lucas V, Tartar A, Davioud-Charvet E. Glutathione-dependent activities of Trypanosoma cruzi p52 makes it a new member of the thiol:disulphide oxidoreductase family. Biochem J. 1997 Feb 15; 322 ( Pt 1):43-8. PMID: 9078241.
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    56. Zoukhri D, Hodges RR, Sergheraert C, Toker A, Dartt DA. Lacrimal gland PKC isoforms are differentially involved in agonist-induced protein secretion. Am J Physiol. 1997 Jan; 272(1 Pt 1):C263-9. PMID: 9038832.
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    57. Loing E, Delanoye A, Sergheraert C, Tartar A, Gras-Masse H. Assessing delivery of lipopeptides into the cytoplasm of intact cells by a functional assay based on PKC inhibition. I. The Jurkat model. Pept Res. 1996 Sep-Oct; 9(5):229-32. PMID: 9000248.
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    58. Baillet S, Buisine E, Horvath D, Maes L, Bonnet B, Sergheraert C. 2-Amino diphenylsulfides as inhibitors of trypanothione reductase: modification of the side chain. Bioorg Med Chem. 1996 Jun; 4(6):891-9. PMID: 8818240.
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    59. Deprez B, Sauzet JP, Boutillon C, Martinon F, Tartar A, Sergheraert C, Guillet JG, Gomard E, Gras-Masse H. Comparative efficiency of simple lipopeptide constructs for in vivo induction of virus-specific CTL. Vaccine. 1996 Apr; 14(5):375-82. PMID: 8735547.
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    60. Ouaissi MA, Dubremetz JF, Schöneck R, Fernandez-Gomez R, Gomez-Corvera R, Billaut-Mulot O, Taibi A, Loyens M, Tartar A, Sergheraert C, et al. Trypanosoma cruzi: a 52-kDa protein sharing sequence homology with glutathione S-transferase is localized in parasite organelles morphologically resembling reservosomes. Exp Parasitol. 1995 Dec; 81(4):453-61. PMID: 8542986.
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    61. Fernandez-Gomez R, Moutiez M, Aumercier M, Bethegnies G, Luyckx M, Ouaissi A, Tartar A, Sergheraert C. 2-Amino diphenylsulfides as new inhibitors of trypanothione reductase. Int J Antimicrob Agents. 1995 Dec; 6(2):111-8. PMID: 18611694.
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    62. Moutiez M, Aumercier M, Parmentier B, Tartar A, Sergheraert C. Compared recognition of di- and trisulfide substrates by glutathione and trypanothione reductases. Biochim Biophys Acta. 1995 Oct 19; 1245(2):161-6. PMID: 7492572.
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    63. Moutiez M, Aumercier M, Schöneck R, Meziane-Cherif D, Lucas V, Aumercier P, Ouaissi A, Sergheraert C, Tartar A. Purification and characterization of a trypanothione-glutathione thioltransferase from Trypanosoma cruzi. Biochem J. 1995 Sep 01; 310 ( Pt 2):433-7. PMID: 7654179.
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    64. Hussain R, Sergheraert C, Drake AF, Siligardi G. Structure-activity relationships and physico-chemical properties of synthetic lipopeptide inhibitors of PKC. Biomed Pept Proteins Nucleic Acids. 1995; 1(2):69-72. PMID: 9346856.
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    65. Meziane-Cherif D, Aumercier M, Kora I, Sergheraert C, Tartar A, Dubremetz JF, Ouaissi MA. Trypanosoma cruzi: immunolocalization of trypanothione reductase. Exp Parasitol. 1994 Dec; 79(4):536-41. PMID: 8001664.
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    66. Aumercier M, Meziane-Cherif D, Moutiez M, Tartar A, Sergheraert C. A microplate assay for trypanothione reductase inhibitors. Anal Biochem. 1994 Nov 15; 223(1):161-4. PMID: 7695093.
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    67. Moutiez M, Aumercier M, Teissier E, Parmentier B, Tartar A, Sergheraert C. Reduction of a trisulfide derivative of glutathione by glutathione reductase. Biochem Biophys Res Commun. 1994 Aug 15; 202(3):1380-6. PMID: 8060317.
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    68. Sqalli-Houssaini H, Pierlot C, Kusnierz JP, Parmentier B, Martin-Nizard F, Lestavel-Delattre S, Tartar A, Fruchart JC, Sergheraert C, Duriez P. Preparation of anti-HIV-low-density lipoprotein complexes for delivery of anti-HIV drugs via the low-density lipoprotein pathways. Biotechnol Ther. 1994; 5(1-2):69-85. PMID: 7703834.
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    69. Sergheraert C, Pierlot C, Tartar A, Henin Y, Lemaitre M. Synthesis and anti-HIV evaluation of D4T and D4T 5'-monophosphate prodrugs. J Med Chem. 1993 Apr 02; 36(7):826-30. PMID: 8385224.
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    70. Zoukhri D, Sergheraert C, Rossignol B. Phorbol ester-stimulated exocytosis in lacrimal gland: PKC might not be the sole effector. Am J Physiol. 1993 Apr; 264(4 Pt 1):C1045-50. PMID: 8386449.
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    71. Zoukhri D, Pelosin JM, Mauduit P, Chambaz E, Sergheraert C, Rossignol B. The rat lacrimal gland expresses the alpha isoform of PKC. Further evidence for the PMA-activated and phospholipid-independent protein kinase activity. Cell Signal. 1992 Jan; 4(1):111-9. PMID: 1571202.
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    72. Pelosin JM, Ricouart A, Sergheraert C, Benahmed M, Chambaz EM. Expression of protein kinase C isoforms in various steroidogenic cell types. Mol Cell Endocrinol. 1991 Feb; 75(2):149-55. PMID: 2050274.
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    73. Ricouart A, Gesquiere JC, Tartar A, Sergheraert C. Design of potent protein kinase inhibitors using the bisubstrate approach. J Med Chem. 1991 Jan; 34(1):73-8. PMID: 1992155.
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    74. Ricouart A, Tartar A, Sergheraert C. Inhibition of protein kinase C by retro-inverso pseudosubstrate analogues. Biochem Biophys Res Commun. 1989 Dec 29; 165(3):1382-90. PMID: 2514686.
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    75. Ricouart A, Tartar A, Sergheraert C. Evidence for negative control in protein kinase C substrate specificity. Int J Pept Protein Res. 1989 Apr; 33(4):304-7. PMID: 2753600.
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    76. Ricouart A, Maes P, Battmann T, Kerdelhue B, Tartar A, Sergheraert C. Photosubstitution of cymantrenylalanine as a tool in peptide chemistry. Synthesis and biological activity of new GnRH analogs. Int J Pept Protein Res. 1988 Jul; 32(1):56-63. PMID: 3065262.
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